商品信息
联系客服
郑重提醒:
无质量问题不接受退换货,下单前请仔细核对信息。
下单后请及时联系客服核对商品价格,订单生效后再付款。
Description:Potent,selectiveCysLT1(LTD4)antagoNIST;orallyactive
AlternativeNames:Ro24-5913
ChemicalName:4-[[3-[(1E)-2-(4-Cyclobutyl-2-thiazolyl)ethenyl]phenyl]amino]-2,2-diethyl-4-oxobutanoicacid
Purity:≥98%(HPLC)
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences
BiologicalActivity
Potent,selectiveCysLT1(LTD4)leukotrienereceptorantagonist(IC50=6.4nM).InhibitsLTD4-inducedbronchoconstrictioninguineapigswhenadministeredintravenously,orallyorbyaerosol.
CompoundLibraries
CinalukastisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
M.Wt | 412.55 |
Formula | C23H28N2O3S |
Storage | Desiccateat-20°C |
Purity | ≥98%(HPLC) |
CASNumber | 128312-51-6 |
PubChemID | 6436135 |
InChIKey | BZMKNPGKXJAIDV-VAWYXSNFSA-N |
Smiles | CCC(CC)(CC(=O)NC1=CC(C=CC2=NC(=CS2)C2CCC2)=CC=C1)C(O)=O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
Solvent | MaxConc.mg/mL | MaxConc.mM | |
---|---|---|---|
Solubility | |||
DMSO | 41.26 | 100 | |
ethanol | 4.13 | 10 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight412.55.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|---|---|---|
1mM | 2.42mL | 12.12mL | 24.24mL |
5mM | 0.48mL | 2.42mL | 4.85mL |
10mM | 0.24mL | 1.21mL | 2.42mL |
50mM | 0.05mL | 0.24mL | 0.48mL |
MolarityCalculator
MolarityCalculator
Calculatethemass,volume,orconcentrationrequiredforasolution.
ReconstitutionCalculator
ReconstitutionCalculator
DilutionCalculator
DilutionCalculator
Calculatethedilutionrequiredtoprepareastocksolution.
ProductDatasheets
CertificateofAnalysis/ProductDatasheet
SafetyDatasheet
▍
品牌分类
▍
官网分类
▍
品牌问答
暂无品牌问答